{"id":60703,"date":"2022-10-27T09:18:39","date_gmt":"2022-10-27T08:18:39","guid":{"rendered":"https:\/\/www.kalapa-clinic.com\/?p=60703"},"modified":"2022-10-27T11:38:29","modified_gmt":"2022-10-27T10:38:29","slug":"raphael-mechoulam-le-pionnier-du-cannabis-medicinal","status":"publish","type":"post","link":"https:\/\/www.kalapa-clinic.com\/fr\/raphael-mechoulam-le-pionnier-du-cannabis-medicinal\/","title":{"rendered":"Raphael Mechoulam: Le pionnier du cannabis m\u00e9dicinal"},"content":{"rendered":"\n<p class=\"wp-block-paragraph\"><strong>Il est l&rsquo;un des plus grands de la chimie pharmaceutique : Le scientifique isra\u00e9lien Raphael Mechoulam est consid\u00e9r\u00e9 comme le d\u00e9couvreur des principes actifs essentiels de la plante de cannabis et de leurs structures chimiques, ainsi que du fonctionnement du syst\u00e8me endocannabino\u00efde humain. Le chercheur, aujourd&rsquo;hui \u00e2g\u00e9 de 91 ans, revient sur une vie mouvement\u00e9e, tant sur le plan personnel que dans son r\u00f4le de scientifique.<\/strong><\/p>\n\n\n\n<h2 class=\"wp-block-heading\">L&rsquo;enfance dans les Balkans<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">Raphael Mechoulam est n\u00e9 \u00e0 Sofia, en Bulgarie, en 1930. Son p\u00e8re, consid\u00e9r\u00e9 comme un m\u00e9decin respect\u00e9, \u00e9tait le directeur de l&rsquo;h\u00f4pital juif local. Raphael a fr\u00e9quent\u00e9 une \u00e9cole primaire am\u00e9ricaine \u00e0 Sofia pendant la premi\u00e8re moiti\u00e9 de son enfance et a pass\u00e9 la seconde en exil : apr\u00e8s la menace nazie, la famille Mechoulam s&rsquo;est cach\u00e9e dans divers villages des Balkans.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Le p\u00e8re a \u00e9t\u00e9 emmen\u00e9 dans un camp de concentration en 1944, mais a heureusement surv\u00e9cu \u00e0 la captivit\u00e9.<\/p>\n\n\n\n<h2 class=\"wp-block-heading\">\u00c9migration vers Isra\u00ebl<\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">Apr\u00e8s la fin de la Seconde Guerre mondiale, la famille Mechoulam a \u00e9migr\u00e9 en Isra\u00ebl. Raphael Mechoulam \u00e9tudie la biochimie \u00e0 l&rsquo;Universit\u00e9 h\u00e9bra\u00efque de J\u00e9rusalem et obtient son doctorat en 1958. De 1953 \u00e0 1955, il s&rsquo;\u00e9tait consacr\u00e9 \u00e0 la recherche sur les insecticides dans le cadre de ses travaux de recherche m\u00e9dicale au service militaire.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Apr\u00e8s avoir obtenu son doctorat, il obtient un poste postdoctoral \u00e0 l&rsquo;Institut Rockefeller de New York mais revient \u00e0 J\u00e9rusalem d\u00e8s 1960. <strong>C&rsquo;est l\u00e0, \u00e0 l&rsquo;Institut Weizmann, que commence la voie de recherche la plus importante de la vie de Mechoulam : l&rsquo;\u00e9tude des principes actifs de la plante de cannabis.<\/strong>&nbsp;<\/p>\n\n\n\n<h2 class=\"wp-block-heading\"><strong>Carri\u00e8re scientifique<\/strong><\/h2>\n\n\n\n<p class=\"wp-block-paragraph\">\u00c0 partir de 1966, Mechoulam a travaill\u00e9 \u00e0 l&rsquo;universit\u00e9 h\u00e9bra\u00efque de J\u00e9rusalem, d&rsquo;abord en tant que scientifique, puis en tant que professeur et recteur de l&rsquo;universit\u00e9. Dans les ann\u00e9es 1990, des visites de recherche et des postes de professeur invit\u00e9 l&rsquo;ont conduit aux \u00c9tats-Unis ; Mechoulam a \u00e9galement \u00e9t\u00e9 pr\u00e9sident de la \u00ab\u00a0International Cannabinoid Research Society\u00a0\u00bb de 1999 \u00e0 2000. <strong>Il a re\u00e7u de nombreux prix, dont le \u00ab\u00a0Prix isra\u00e9lien des sciences exactes\u00a0\u00bb (2000) et le prestigieux prix Harvey, consid\u00e9r\u00e9 comme un pr\u00e9curseur du prix Nobel (2020).<\/strong> Ce dernier a \u00e9t\u00e9 d\u00e9cern\u00e9 en reconnaissance des d\u00e9couvertes pionni\u00e8res de Mechoulam dans le domaine du cannabis m\u00e9dicinal.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Mechoulam vit toujours \u00e0 J\u00e9rusalem et est toujours consid\u00e9r\u00e9 comme le plus important pionnier de la recherche sur le cannabis.<\/p>\n\n\n\n<h2 class=\"wp-block-heading\">Les grandes \u00e9tapes de la recherche sur les cannabino\u00efdes : Les m\u00e9rites de Mechoulam<\/h2>\n\n\n\n<h3 class=\"wp-block-heading\">1963\/1964 : D\u00e9couverte du CBD et du THC<\/h3>\n\n\n\n<ul class=\"wp-block-list\"><li>L&rsquo;\u00e9quipe de Mechoulam obtient cinq kilos de \u00ab\u00a0haschisch\u00a0\u00bb n\u00e9cessaires \u00e0 la recherche dans la salle des preuves d&rsquo;un poste de police isra\u00e9lien &#8211; vraisemblablement une saisie de contrebande en provenance du Liban.<\/li><li>Isolation du cannabidiol (CBD), l&rsquo;un des centaines de compos\u00e9s actifs du chanvre, et description de sa structure chimique. Un an plus tard, isolement du composant psychotrope t\u00e9trahydrocannabinol (THC), responsable de l&rsquo;effet intoxicant du cannabis.<\/li><\/ul>\n\n\n\n<p class=\"wp-block-paragraph\">Premi\u00e8re publication de l&rsquo;\u00e9quipe de recherche sur l&rsquo;effet th\u00e9rapeutique du CBD dans les maladies suivantes&nbsp;:<\/p>\n\n\n\n<ul class=\"wp-block-list\"><li>Inflammation<\/li><li>l&rsquo;anxi\u00e9t\u00e9<\/li><li>le diab\u00e8te de type 1<\/li><li>Maladies auto-immunes<\/li><li>Maladies neurologiques<\/li><\/ul>\n\n\n\n<h3 class=\"wp-block-heading\">Fin des ann\u00e9es 60\/d\u00e9but des ann\u00e9es 70 : Recherche sur les singes<\/h3>\n\n\n\n<ul class=\"wp-block-list\"><li>Test des effets des principaux cannabino\u00efdes \u00e0 base de plantes sur les singes. Reconfirmation : Le THC a des effets psychotropes sur les singes, mais pas le CBD.<\/li><\/ul>\n\n\n\n<h3 class=\"wp-block-heading\">1980 : Premi\u00e8re \u00e9tude en double aveugle sur les effets du CBD dans l&rsquo;\u00e9pilepsie.<\/h3>\n\n\n\n<ul class=\"wp-block-list\"><li>D\u00e9but des recherches sur les effets du CBD et du THC sur l&rsquo;\u00e9pilepsie &#8211; d&rsquo;abord sur des souris. Par la suite, une \u00e9tude en double aveugle sur l&rsquo;effet du CBD chez des patients \u00e9pileptiques pr\u00e9sentant des sympt\u00f4mes chroniques a donn\u00e9 des r\u00e9sultats impressionnants : Apr\u00e8s trois mois de traitement au CBD, les crises ont \u00e9t\u00e9 \u00e9limin\u00e9es ou r\u00e9duites de mani\u00e8re significative.<\/li><li>Les r\u00e9sultats de l&rsquo;\u00e9tude n&rsquo;ont pas suscit\u00e9 un grand int\u00e9r\u00eat dans le monde de la recherche ou sur les march\u00e9s pharmaceutiques, probablement en raison de la stigmatisation attach\u00e9e au cannabis.<\/li><\/ul>\n\n\n\n<h3 class=\"wp-block-heading\">1992 : D\u00e9voilement du syst\u00e8me endocannabino\u00efde (ECS)<\/h3>\n\n\n\n<ul class=\"wp-block-list\"><li>Identification des endocannabino\u00efdes anandamide et 2-arachidonylglyc\u00e9ro (2-AG), que le corps humain produit lui-m\u00eame et qui interagissent avec les r\u00e9cepteurs CB1 et CB2.<\/li><\/ul>\n\n\n\n<ul class=\"wp-block-list\"><li>L&rsquo;\u00e9quipe de recherche a observ\u00e9 des interactions similaires par l&rsquo;administration externe de cannabino\u00efdes et a ainsi d\u00e9couvert le syst\u00e8me cannabino\u00efde endog\u00e8ne, \u00e9galement appel\u00e9 syst\u00e8me endocannabino\u00efde (SEC).<\/li><li>La connaissance du fonctionnement du syst\u00e8me endocannabino\u00efde est \u00e0 la base de l&rsquo;utilisation th\u00e9rapeutique actuelle du Cannabis sativa et des principes actifs de la plante.<\/li><\/ul>\n\n\n\n<h3 class=\"wp-block-heading\">2002 : Recherche sur les l\u00e9sions c\u00e9r\u00e9brales traumatiques<\/h3>\n\n\n\n<ul class=\"wp-block-list\"><li>D\u00e9couverte d&rsquo;une production accrue d&rsquo;anandamide et de 2-AG dans le cerveau apr\u00e8s une l\u00e9sion c\u00e9r\u00e9brale traumatique. En outre, les deux endocannabino\u00efdes produits par l&rsquo;organisme inhibent la production de substances nocives apr\u00e8s une l\u00e9sion intracr\u00e2nienne.<\/li><li>\u00c9tude du potentiel inhibiteur de l&rsquo;anandamide et du 2-AG dans les l\u00e9sions neuronales apr\u00e8s une l\u00e9sion c\u00e9r\u00e9brale traumatique chez la souris et le rat : L&rsquo;administration de ces compos\u00e9s r\u00e9duit de mani\u00e8re significative l&rsquo;\u00e9tendue des l\u00e9sions c\u00e9r\u00e9brales.<\/li><\/ul>\n\n\n\n<p class=\"wp-block-paragraph\"><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Nous sommes particuli\u00e8rement reconnaissants au Professeur Mechoulam d&rsquo;avoir fourni la photo pour cet article.<\/p>\n\n\n\n<p class=\"wp-block-paragraph\"><strong>Sources:<\/strong><\/p>\n\n\n\n<p class=\"wp-block-paragraph\">Mechoulam, R. (2022). A Delightful Trip Along the Pathway of Cannabinoid and Endocannabinoid Chemistry and Pharmacology. <em>Annual Review of Pharmacology and Toxicology<\/em>, <em>63<\/em>(1). <a href=\"https:\/\/doi.org\/10.1146\/annurev-pharmtox-051921-083709\">https:\/\/doi.org\/10.1146\/annurev-pharmtox-051921-083709<\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Il est l&rsquo;un des plus grands de la chimie pharmaceutique : Le scientifique isra\u00e9lien Raphael Mechoulam est consid\u00e9r\u00e9 comme le d\u00e9couvreur des principes actifs essentiels de la plante de cannabis et de leurs structures chimiques, ainsi que du fonctionnement du syst\u00e8me endocannabino\u00efde humain. Le chercheur, aujourd&rsquo;hui \u00e2g\u00e9 de 91 ans, revient sur une vie mouvement\u00e9e, [&#8230;]<\/p>\n<p><a class=\"understrap-read-more-link\" href=\"https:\/\/www.kalapa-clinic.com\/fr\/raphael-mechoulam-le-pionnier-du-cannabis-medicinal\/\">En savoir plus \u2192<\/a><\/p>\n","protected":false},"author":48,"featured_media":60846,"comment_status":"closed","ping_status":"closed","sticky":false,"template":"","format":"standard","meta":{"inline_featured_image":false,"_uag_custom_page_level_css":"","footnotes":""},"categories":[5106,5098,5099],"tags":[4686,4648,4650,4696,4691,4685],"class_list":["post-60703","post","type-post","status-publish","format-standard","has-post-thumbnail","hentry","category-actualites-cannabis","category-aktuelle-nachrichten","category-latest-news","tag-anxiete","tag-cannabis-medical","tag-cannabis-therapeutique","tag-plante-de-cannabis","tag-systeme-endocannabinoide","tag-traitement-aux-cannabinoides"],"yoast_head":"<!-- This site is optimized with the 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